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MCL1 - Mcl1 Protein

- July 29, 2017

BH3 domain-independent apolipoprotein L1 toxicity rescued by BCL2 ...
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Induced myeloid leukemia cell differentiation protein Mcl-1 is a protein that in humans is encoded by the MCL1 gene.


Vanderbilt Institute of Chemical Biology
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Function

The protein encoded by this gene belongs to the Bcl-2 family. Alternative splicing occurs at this locus and two transcript variants encoding distinct isoforms have been identified. The longer gene product (isoform 1) enhances cell survival by inhibiting apoptosis while the alternatively spliced shorter gene product (isoform 2) promotes apoptosis and is death-inducing.


Mcl1 Protein Video



Clinical significance

Omacetaxine mepesuccinate (a drug approved for the treatment for chronic myelogenous leukemia (CML)) and Seliciclib (which is under investigation as a potential multiple myeloma treatment) both act in part by inhibiting synthesis of Mcl-1.


Gain-of-function microRNA screens identify miR-193a regulating ...
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Interactions

MCL1 has been shown to interact with:

  • BAK1,
  • BCL2L11,
  • BID,
  • BAD,
  • DAD1,
  • PMAIP1,
  • PCNA,
  • TCTP and
  • TNKS

Source of the article : Wikipedia



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